Mutations in SLC6A1, encoding γ-aminobutyric acid (GABA) transporter 1 (GAT-1), have been recently associated with a spectrum of epilepsy syndromes, intellectual disability and autism in clinic. However, the pathophysiology of the gene mutations is far from clear.
Here we report a novel SLC6A1 missense mutation in a patient with epilepsy and autism spectrum disorder and characterized the molecular defects of the mutant GAT-1, from transporter protein trafficking to GABA uptake function in heterologous cells and neurons. The heterozygous missense mutation (c1081C to A (P361T)) in SLC6A1 was identified by exome sequencing. We have thoroughly characterized the molecular pathophysiology underlying the clinical phenotypes. We performed EEG recordings and autism diagnostic interview.
Mac-2BP Polyclonal Antibody |
ABP59179-01ml |
Abbkine |
0.1ml |
EUR 289 |
|
Description: A polyclonal antibody for detection of Mac-2BP from Human, Mouse. This Mac-2BP antibody is for WB, ELISA. It is affinity-purified from rabbit serum by affinity-chromatography using the specific immunogenand is unconjugated. The antibody is produced in rabbit by using as an immunogen synthesized peptide derived from part region of human Mac-2BP protein at amino acid sequence of 100-160 |
Mac-2BP Polyclonal Antibody |
ABP59179-02ml |
Abbkine |
0.2ml |
EUR 414 |
|
Description: A polyclonal antibody for detection of Mac-2BP from Human, Mouse. This Mac-2BP antibody is for WB, ELISA. It is affinity-purified from rabbit serum by affinity-chromatography using the specific immunogenand is unconjugated. The antibody is produced in rabbit by using as an immunogen synthesized peptide derived from part region of human Mac-2BP protein at amino acid sequence of 100-160 |
Anti-Mac-2BP antibody |
STJ98720 |
St John's Laboratory |
200 µl |
EUR 197 |
Description: Rabbit polyclonal to Mac-2BP. |
Mac-2BP Polyclonal Antibody |
46771-100ul |
SAB |
100ul |
EUR 252 |
Mac-2BP Polyclonal Antibody |
46771-50ul |
SAB |
50ul |
EUR 187 |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC040271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF405S conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC040271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF405S conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC470271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF647 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC470271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF647 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC550271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF555 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC550271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF555 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNCB0271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),Biotin conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNCB0271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),Biotin conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC810271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF680R conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC810271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF680R conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC700271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF770 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC700271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF770 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC880271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF488A conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC880271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF488A conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC940271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF594 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC940271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF594 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC680271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF568 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC680271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF568 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNCA0271-250 |
Biotium |
250uL |
EUR 383 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),APC conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNCAP0271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),Alkaline Phosphatase conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNCAP0271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),Alkaline Phosphatase conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNUM0271-50 |
Biotium |
50uL |
EUR 395 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271), 1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNCP0271-250 |
Biotium |
250uL |
EUR 383 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),PerCP conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC050271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF405M conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC050271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF405M conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC400271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF640R conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC400271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF640R conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNCR0271-250 |
Biotium |
250uL |
EUR 383 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),RPE conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNUB0271-100 |
Biotium |
100uL |
EUR 209 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271), Concentration: 0.2mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNUB0271-500 |
Biotium |
500uL |
EUR 458 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271), Concentration: 0.2mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC430271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF543 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC430271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF543 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNCH0271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),Horseradish Peroxidase conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNCH0271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),Horseradish Peroxidase conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC610271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF660R conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC610271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF660R conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC800271-100 |
Biotium |
100uL |
EUR 199 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF680 conjugate, Concentration: 0.1mg/mL |
CD11b / MAC-1 (Microglial Marker) (ITGAM/271) Antibody |
BNC800271-500 |
Biotium |
500uL |
EUR 544 |
Description: Primary antibody against CD11b / MAC-1 (Microglial Marker) (ITGAM/271),CF680 conjugate, Concentration: 0.1mg/mL |
Mac-2BP Polyclonal Conjugated Antibody |
C46771 |
SAB |
100ul |
EUR 397 |
Recombinant H9N2 MAC Hemagglutinin / HA Protein (aa 1-523) [His] |
VAng-Wyb6928-100g |
Creative Biolabs |
100 µg |
EUR 1741 |
Description: Influenza A H9N2 (A/Chicken/Hong Kong/G9/97) Hemagglutinin / HA, recombinant protein. |
Recombinant H9N2 MAC Hemagglutinin / HA Protein (aa 1-523) [His] |
VAng-Wyb6928-50g |
Creative Biolabs |
50 µg |
EUR 1050 |
Description: Influenza A H9N2 (A/Chicken/Hong Kong/G9/97) Hemagglutinin / HA, recombinant protein. |
Human membrane attack complex(MAC)ELISA Kit |
GA-E0376HM-48T |
GenAsia Biotech |
48T |
EUR 289 |
Human membrane attack complex(MAC)ELISA Kit |
GA-E0376HM-96T |
GenAsia Biotech |
96T |
EUR 466 |
Human membrane attack complex,MAC ELISA Kit |
201-12-0360 |
SunredBio |
96 tests |
EUR 440 |
|
Description: A quantitative ELISA kit for measuring Human in samples from biological fluids. |
Human Membrane Attack Complex (MAC) ELISA Kit |
abx350654-96tests |
Abbexa |
96 tests |
EUR 668 |
|
Human membrane attack complex,MAC ELISA Kit |
CN-04250H1 |
ChemNorm |
96T |
EUR 442 |
Human membrane attack complex,MAC ELISA Kit |
CN-04250H2 |
ChemNorm |
48T |
EUR 293 |
Polyclonal Integrin alpha-M (CD11b, MAC-1, OX-42 Antigen) Antibody |
AMM06021G |
Leading Biology |
0.1mg |
EUR 528 |
Description: A polyclonal antibody raised in Chicken that recognizes and binds to Human Integrin alpha-M (CD11b, MAC-1, OX-42 Antigen) . This antibody is tested and proven to work in the following applications: |
Recombinant H9N2 MAC Hemagglutinin HA1 Subunit Protein (aa 1-338) [His] |
VAng-Wyb6929-100g |
Creative Biolabs |
100 µg |
EUR 1741 |
Description: Influenza A H9N2 (A/Chicken/Hong Kong/G9/97) Hemagglutinin HA1 Subunit, recombinant protein. |
Recombinant H9N2 MAC Hemagglutinin HA1 Subunit Protein (aa 1-338) [His] |
VAng-Wyb6929-10g |
Creative Biolabs |
10 µg |
EUR 573 |
Description: Influenza A H9N2 (A/Chicken/Hong Kong/G9/97) Hemagglutinin HA1 Subunit, recombinant protein. |
Recombinant H9N2 MAC Hemagglutinin HA1 Subunit Protein (aa 1-338) [His] |
VAng-Wyb6929-50g |
Creative Biolabs |
50 µg |
EUR 1050 |
Description: Influenza A H9N2 (A/Chicken/Hong Kong/G9/97) Hemagglutinin HA1 Subunit, recombinant protein. |
ELISA kit for Human MAC (Membrane Attack Complex) |
E-EL-H5418 |
Elabscience Biotech |
1 plate of 96 wells |
EUR 534 |
|
Description: A sandwich ELISA kit for quantitative measurement of Human MAC (Membrane Attack Complex) in samples from Serum, Plasma, Cell supernatant |
ELISA kit for Human Membrane attack complex (MAC) |
KTE62641-48T |
Abbkine |
48T |
EUR 354 |
|
Description: Quantitative sandwich ELISA for measuring Human Membrane attack complex (MAC) in samples from cell culture supernatants, serum, whole blood, plasma and other biological fluids. |
ELISA kit for Human Membrane attack complex (MAC) |
KTE62641-5platesof96wells |
Abbkine |
5 plates of 96 wells |
EUR 2252 |
|
Description: Quantitative sandwich ELISA for measuring Human Membrane attack complex (MAC) in samples from cell culture supernatants, serum, whole blood, plasma and other biological fluids. |
ELISA kit for Human Membrane attack complex (MAC) |
KTE62641-96T |
Abbkine |
96T |
EUR 572 |
|
Description: Quantitative sandwich ELISA for measuring Human Membrane attack complex (MAC) in samples from cell culture supernatants, serum, whole blood, plasma and other biological fluids. |
Monoclonal CD11b / MAC-1 (Microglial Marker) Antibody - With BSA and Azide, Clone: M1/70 |
AMM05473G |
Leading Biology |
0.05mg |
EUR 396 |
Description: A Monoclonal antibody against Human CD11b / MAC-1 (Microglial Marker) - With BSA and Azide. The antibodies are raised in Rat and are from clone M1/70. This antibody is applicable in IHC, IF, FC, IP, E |
Monoclonal CD11b / MAC-1 (Microglial Marker) Antibody - With BSA and Azide, Clone: C11b/660 |
APG03040G |
Leading Biology |
0.05mg |
EUR 396 |
Description: A Monoclonal antibody against Human CD11b / MAC-1 (Microglial Marker) - With BSA and Azide. The antibodies are raised in Mouse and are from clone C11b/660. This antibody is applicable in IHC, IF, FC, IP, E |
Monoclonal CD11b / MAC-1 (Microglial Marker) Antibody - Without BSA and Azide, Clone: M1/70 |
APG03041G |
Leading Biology |
0.1mg |
EUR 484 |
Description: A Monoclonal antibody against Human CD11b / MAC-1 (Microglial Marker) - Without BSA and Azide. The antibodies are raised in Rat and are from clone M1/70. This antibody is applicable in IF, FC |
Monoclonal CD11b / MAC-1 (Microglial Marker) Antibody - Without BSA and Azide, Clone: C11b/660 |
APG03042G |
Leading Biology |
0.1mg |
EUR 484 |
Description: A Monoclonal antibody against Human CD11b / MAC-1 (Microglial Marker) - Without BSA and Azide. The antibodies are raised in Mouse and are from clone C11b/660. This antibody is applicable in IF, FC |
Monoclonal MAC-2-BP / LGALS3BP Antibody (clone 2B1), Clone: 2B1 |
AMM02212G |
Leading Biology |
0.05ml |
EUR 484 |
Description: A Monoclonal antibody against Human MAC-2-BP / LGALS3BP (clone 2B1). The antibodies are raised in Mouse and are from clone 2B1. This antibody is applicable in WB and IHC-P, Flo |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, GST, E.coli-100ug |
QP5791-ec-100ug |
EnQuireBio |
100ug |
EUR 408 |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, GST, E.coli-10ug |
QP5791-ec-10ug |
EnQuireBio |
10ug |
EUR 200 |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, GST, E.coli-1mg |
QP5791-ec-1mg |
EnQuireBio |
1mg |
EUR 1632 |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, GST, E.coli-200ug |
QP5791-ec-200ug |
EnQuireBio |
200ug |
EUR 634 |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, GST, E.coli-500ug |
QP5791-ec-500ug |
EnQuireBio |
500ug |
EUR 1060 |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, GST, E.coli-50ug |
QP5791-ec-50ug |
EnQuireBio |
50ug |
EUR 263 |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, His, Yeast-100ug |
QP5791-ye-100ug |
EnQuireBio |
100ug |
EUR 480 |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, His, Yeast-10ug |
QP5791-ye-10ug |
EnQuireBio |
10ug |
EUR 236 |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, His, Yeast-1mg |
QP5791-ye-1mg |
EnQuireBio |
1mg |
EUR 1885 |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, His, Yeast-200ug |
QP5791-ye-200ug |
EnQuireBio |
200ug |
EUR 744 |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, His, Yeast-500ug |
QP5791-ye-500ug |
EnQuireBio |
500ug |
EUR 1206 |
Recombinant Human CD59/ CD59A/ MAC-IP Protein, His, Yeast-50ug |
QP5791-ye-50ug |
EnQuireBio |
50ug |
EUR 299 |
Neuregulin/Heregulin-1? (NRG-1?/HRG-1?), human recombinant protein |
P1054-1 |
ApexBio |
1 mg |
EUR 3947 |
Description: Neuregulin (NRG) is a signaling protein for ErbB2/ErbB4 receptor heterodimers on the cardiac muscle cells and plays an important role in heart structure and function through inducing cardiomyocyte differentiation |
Angiotensin 1/2 (1-7) amide |
A1054-1 |
ApexBio |
1 mg |
EUR 96 |
Description: Angiotensin I/II (1-7) amide (H2N-Asp-Arg-Val-Tyr-Ile-His-Pro-amide) is a peptide analog to angiotensin II that is used as a vasopressor in the treatment of certain types of shock and circulatory collapse. |
Angiotensin 1/2 (1-8) amide |
A1055-1 |
ApexBio |
1 mg |
EUR 96 |
Description: The physiologically active peptide angiotensin-2 (angiotensin 1- 8) is yielded from angiotensin-1, a substrate of ACE (angiotensin converting enzyme), by removing a dipeptide. |
Endothelin-1 (1-15), amide, human |
A1111-1 |
ApexBio |
1 mg |
EUR 722 |
Description: Endothelins are 21-amino acid vasoconstricting peptides produced primarily in the endothelium and have a key role in vascular homeostasis. |
Haptoglobin, (Phenotype 1-1) Human Plasma |
7536-1 |
Biovision |
|
EUR 321 |
Flutax 1 |
B6986-1 |
ApexBio |
1 mg |
EUR 399 |
TAPI-1 |
B4686-1 |
ApexBio |
1 mg |
EUR 268 |
Description: TAPI-1 is an inhibitor of tumour necrosis factor with IC50 value of 8.09 ?M [1].TAPI-1 is an inhibitor of TACE/ADAM17 which catalyzes the cleavage of full-length APP to the soluble N-terminal fragment (sAPP?). |
C14TKL-1 |
B5240-1 |
ApexBio |
1 mg |
EUR 399 |
?1-MSH |
B5427-1 |
ApexBio |
1 mg |
EUR 268 |
CRSP-1 |
B5452-.1 |
ApexBio |
100 ug |
EUR 415 |
ADWX 1 |
B5722-.1 |
ApexBio |
100 ug |
EUR 583 |
Description: ADWX 1 is a potent and selective inhibitor of KV1.3 channel with IC50 values of 1.89 pM and 0.65 nM for Kv1.3 and Kv1.1, respectively [1]. |
Purotoxin 1 |
B5771-.1 |
ApexBio |
100 µg |
EUR 380 |
Psalmotoxin 1 |
B5796-.1 |
ApexBio |
100 ug |
EUR 447 |
Description: IC50: 0.9 nMPsalmotoxin 1 is a potent and selective acid-sensing ion channel 1a (ASIC1a) blocker.Several ASIC subunits described: ASIC1a, ASIC1b, ASIC2a, ASIC2b, and ASIC3 with different kinetics, tissue distribution, and external pH sensitivities. |
UK 1 |
C5006-1 |
ApexBio |
1 mg |
EUR 363 |
Description: UK 1, an unusual bis-benzoxazole metabolite isolated from Streptomyces sp. 517-02, is an inhibitor of topoisomerase II (Topo II) and hepatitis C viral replication. |
KP372-1 |
C5053-1 |
ApexBio |
1 mg |
EUR 132 |
Description: IC50: 30-60 nM for thyroid cancer cells KP372-1 is a specific Akt inhibitor. The phosphatidylinositol 3' kinase (PI3K)/phosphatase, which is a key regulator of cell proliferation and survival, is mutated or activated in various cancers. |